NUDIKAULINE PERCHLORATE - LATOXAN Technical Data Sheet
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L6037 NUDIKAULINE PERCHLORATE

aBungarotoxin neuronal nicotinic receptor antagonist with a selectivity comparable to that of Methyllycaconitine at the brain sites (nanomolar affinity); potent medium-acting non depolarizing neuromuscular blocker; muscle relaxant.

  1. see annexed table : Evaluation of 8 Alkaloids for Activity at Neuronal...

Alkaloid C38H50N2O11.HClO4 from plants of the Ranunculaceae family.


PRICES
QuantityUS DollarsEURO
5 mg 141.40 101.00
25 mg 565.60 404.00


  • Molecular Weight : 810.5 Da.

  • Melting Point : 209-212 °C.

  • Solubility in : ethanol.

  • Purity min. : 96% (TLC, mass-spectrometry).

  • Biological Activity : recent studies (see attached sheet) show that Nudikauline perchlorate acts as neuronal a-Bungarotoxin-sensitive brain nicotinic receptors antagonist, with a comparable affinity to Methyllycaconitine.

  • Toxicity (LD50) : mice (i.v.): 1.8 mg/kg. mice (i.p.): 13.0 mg/kg. mice (orally): 38.0 mg/kg.

  • Storage recommendations : Store at +4°C, in dark place.

  • CAS Reg. No. : 99815-83-5

  • Bibliography :
    1. Kulanthaivel et al., Heterocycles (1985). 23:2515



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    Revised : 26/04/2007 10:27 - Copyright © Latoxan