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ION CHANNEL and RECEPTOR LIGANDS TOXINS & ALKALOIDS

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| | L9003 MEBICYPHAT
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| PRICES |
| Quantity | US Dollars | EURO |
1 mg | 102.20 | 73.00 |
5 x 1 mg | 408.80 | 292.00 |
- Molecular Weight : 164 Da.
- Melting Point : 249-250 °C.
- Solubility in : well in alcohol and water.
- Purity min. : 95 % (NMR).
- Biological Activity : Cl- channel blocking concentration: IC100 = 500 nM (Lymnaea stagnalis);
experiments with [3H]-labelled GABA-competitive ligands (Muscimol, Flunitrazepam) showed no influence of Mebicyphat up to 10 µM.
- Toxicity (LD50) : mice (i.p.): 32.0 mg/kg.
mice (i.v.): 30.5 mg/kg.
- Storage recommendations : store at room temperature.
- CAS Reg. No. : 1449-89-4
- Bibliography :
- Bellet E. M., Casida J. E., Sciences (1973). 182:1135-1136
- Cooper G. H. et al., Eur. J. Med. Chem. (1978). 13:207-212
- V. I. Fetisov et al., Biol. Membr.(1986) (Russian). 3(5):968-970
- Squires R. F. et al., Mol. Pharmacol. (1983). 23:326-331
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Revised : 26/04/2007 10:27 - Copyright © Latoxan |
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