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Home Page > Alphabetical Index > LK-66

LK-66 Prod. No L9022 - CAS # 36944-86-2
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Product Name LK-66
Product Code L9022
LK-66

C16H20NS2I

Molecular Formula C16H20NS2I
Description

a highly selective M1 Muscarinic receptor antagonist.

Quaternary ammonium salt‚ C16H20NS2I ‚ synthetic.

 
Biological Activity

pIC50 (= -log IC50):M1 (rat brain) = 8.46

M2 (heart) = 5.10

selectivity: [IC50]M2 / [IC50]M1= 2291

data determined by [3H]-QNB binding method‚ Pirenzepine as standard (unpublished).

 
Chemical and Physical Properties
 
CAS No. 36944-86-2 Molecular Weight 417.37 Da.
RTECS Physical Form
Merck Index No (13th Ed.) Melting point 216-218 °C.
PubChem SID Solubility water (heat up)‚ ethanol.
Purity 95 % (NMR). Optical Activity
Toxicity (LD50)
Chemical Names
Storage & Reconstitution Recommendations Store at +4°C‚ in dark place. Solution for use: 10-3 M.
Safety Recommendations
 
Bibliographic References
  1. V. Malyguin et al.; XIII int. symp. Med. Chem. (Paris : 19-24 sept.); Abstr.; 312 (1994).
 
Prices
Code
Quantity
US $
€uro
L9022
1 x 2 mg
96.60
69.00
5 x 2 mg
386.40
276.00
 
External Links PubMed Biomedical Citations From PubMed Toxicology Citations From PubMed PubChem SID

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