L6205 - STROPHANTIDIN 3-Acetate
(Syn. : Acetylstrophanthidin)
(Syn. : Acetylstrophanthidin)
STROPHANTIDIN 3-Acetate | Product ID | L6205 |
| Name | STROPHANTIDIN 3-Acetate |
| Molecular formula | C25H34O7 |
| Description |
It is an ATPase inhibitor and a cardiotonic. Cardiac glycoside , derivative of Strophantidin from plants of the Strophantus genus, Apocynaceae |
| Biological activity | IC50 for cardiac Na+/K+-ATPase inhibition: 0.4 μM; |
Packaging and Prices
| Packaging | Price (€) | Quantité | Buy Now |
|---|---|---|---|
| 10 mg | 82.00 | ||
| 50 mg | 328.00 | ||
| For quotation of big quantities, please Contact us | |||
Product Technical Documents
 | Safety Data Sheet Available on request, please Contact us Ref. SDS_L6205 : unit price : free of charge |
Chemical and Physical Properties
| Product code | L6205 | Molecular weight | 446.53 g/mol |
| Product name | STROPHANTIDIN 3-Acetate | Physical form | |
| CAS No. | 60-38-8 | Melting point | 238-242 °C (decomp.) |
| RTECS | FH5311400 | Solubility | In chloroform Slightly in ethanol Not in water and ether |
| UNIPROT | Optical Activity | [alpha]D + 52° | |
| PubChem SID | |||
| PubChem CID | 261075 | ||
| Purity | > 98% | ||
| Toxicity(LD50) | IVN-RBT LDLo: 550µg/kg | ||
| Chemical Name | 5-beta-Card-20(22)-enolide,19-oxo-3-beta,5,14-trihydroxy-, 3-acetate | ||
| Storage & Reconstitution Recommandations |
Store at +4°C, in dark place; Solution for use: 0.05 %. |
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| Savety Recommandations | For research use only — not intended for food, diagnostic or therapeutic use |
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Bibliographic References
| Product code | L6205 |
| Product name | STROPHANTIDIN 3-Acetate |
- Kai Yuan Yu, "Inhibition of H+-transporting ATPase, Ca2+-transporting ATPase and H+/K+-transporting ATPase by Strophantidin." Biochim. Biophys. Acta (1992). 1159(1):109-112
- Mirsalichova et al., "The thermodynamic essence of the reversible inactivation of Na+/K+ transporting ATPase by various digitalis derivatives is relaxation of enzyme conformational energy." Bioch. Biophys. Acta (1988). 937:335-346
Links
| Product code | L6205 |
| Product name | STROPHANTIDIN 3-Acetate |
| External Links |
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