QUIRESTON-A
Product ID L9037 
Name QUIRESTON-A 
Molecular formula C10H16BrNO
Description

an inhibitor of high-affinity choline uptake (HAChU) in synaptosomes; acetylcholine synthesis inhibitor; weak penetration of biological membranes.


Quinicludine derivative
Biological activity

Cell impermeable inhibitor of high-affinity choline uptake (HAChU). For comparative information see the attached table.
poor penetration of biological membranes.

 Packaging and Prices

Packaging Price (€) Quantité Buy Now
20 mg 530.00

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100 mg 2 120.00

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For quotation of big quantities, please Contact us
 Product Technical Documents
Safety Data Sheet Available on request, please Contact us
Ref. SDS_L9037 : unit price : free of charge
 Chemical and Physical Properties
Product code L9037  Molecular weight 246.14 Da.
Product name QUIRESTON-A  Physical form slightly yellowish crystal powder
CAS No. Melting point 166-168 °C
RTECS Solubility water, ethanol and DMSO.
UNIPROT Optical Activity
PubChem SID    
PubChem CID    
Purity min. 99.5%. (NMR (D2O))    
Toxicity(LD50) mice (orally) 500 mg/kg    
Chemical Name 1-allyl 3-quinicludon bromide; N-allyl-3-oxoquinuclidinium bromide.    
Storage & Reconstitution
Recommandations

Store in a dark place in a dessicator; solutions are stable for 1-2 days at room temperature. Solution for use: 10-3M (2 mg in 8.13 ml).


 
Savety Recommandations  
 Bibliographic References
Product code L9037 
Product name QUIRESTON-A 

- Dahlbom R. et al., "Cell Mol. Basis Cholinergic Funct.", Dowdall M. J. and Hawthorne J. N. Eds., Horwood, Chichester U.K., (1987) 347-354
- Sterling et al., "Inhibition of high-affinity choline uptake and acetylcholine synthesis by quinuclidinyl and hemicholinium derivatives", J. Neurochem.(1986). 46(14):1170-1175
- Doukas P.H. et al., ibid, 355-360
- Baltzod F. et al., Biochem. Pharm. (1980). 29(18):2413-2416
- Tamaru M. et al., Brain Res (1988). 473(2):205-226
- Dowdall M.J. et al., in Cholinergic mechanisms and Psycopharmacology, Ed. D.J.Jenden, Plenum Press, N-Y, (1978). 359
 Links
Product code L9037 
Product name QUIRESTON-A 
External Links PubMed
Biomedical Citations From PubMed
Toxicology Citations From PubMed
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